反应条件
1: triethylamine; palladium diacetate; 9,9-dimethyl-4,5-bis(diphenyl-phosphino)xanthene / N,N-dimethyl-formamide / 12 h / 100 °C 2: lithium hydroxide hydrate; water / tetrahydrofuran; methanol / 3 h / 20 °C View Scheme
参考文献
Journal of Medicinal Chemistry, , vol. 57, # 6 p. 2692 - 2703