反应条件
1.1: triethylamine / N,N-dimethyl-formamide 1.2: 24 h 2.1: pyridine; 4-(N,N-dimethlyamino)pyridine; di-tert-butyl dicarbonate / 24 h 3.1: water; sodium hydroxide / acetone / 1.5 h / -2 °C 3.2: pH 4 View Scheme
参考文献
Cui, Hong-Kui; Guo, Ye; He, Yao; Wang, Feng-Liang; Chang, Hao-Nan; Wang, Yu-Jia; Wu, Fang-Ming; Tian, Chang-Lin; Liu, Lei
Angewandte Chemie - International Edition, 2013 , vol. 52, # 36 p. 9558 - 9562
Angew. Chem., 2013 , vol. 125, # 36 p. 9737 - 9741,5