sodium hydroxide in 1,4-dioxane; water T=0 - 20°C;
参考文献
Gavande, Navnath; Kim, Hye-Lim; Doddareddy, Munikumar R.; Johnston, Graham A. R.; Chebib, Mary; Hanrahan, Jane R.
ACS Medicinal Chemistry Letters, 2013 , vol. 4, # 4 p. 402 - 407
Egbertson, Melissa S.; Chang, Charles T.-C.; Duggan, Mark E.; Gould, Robert J.; Halczenko, Wasyl; et al.
Journal of Medicinal Chemistry, 1994 , vol. 37, # 16 p. 2537 - 2551