反应条件
1: 1,3-thiazole With n-butyllithium in diethyl ether T=-78°C; 0.25 h; 2: N,O-dimethylacetohydroxamic acid in tetrahydrofuran; diethyl ether T=-78 - 20°C;
参考文献
Farmer, Luc J.; Bemis, Guy; Britt, Shawn D.; Cochran, John; Connors, Martin; Harrington, Edmund M.; Hoock, Thomas; Markland, William; Nanthakumar, Suganthini; Taslimi, Paul; Haar, Ernst Ter; Wang, Jian; Zhaveri, Darshana; Salituro, Francesco G.
Bioorganic and Medicinal Chemistry Letters, 2008 , vol. 18, # 23 p. 6231 - 6235