反应条件
1: 1.) NH2OH, NaOH, HCl, 2.) HCl / 1.) MeOH, H2O, -30 deg C, 1.5 h, 0 deg C, 1 h, 2.) H2O, MeOH, 80 deg C, 1 h 2: 60 percent / K2CO3 / acetone / 24 h / 50 °C View Scheme
参考文献
Slok; Ebert; Lang; Krogsgaard-Larsen; Lenz; Madsen
European Journal of Medicinal Chemistry, 1997 , vol. 32, # 4 p. 329 - 338