反应条件
1: HCl / diethyl ether / Heating 2: H2 / PtO2 / ethanol 3: 1.) Na, 3.) conc. HCl 4: 77 percent / 20percent aq. chloroacetic acid, AcOH / 18 h / Heating View Scheme
参考文献
Orr; Musso; Boswell; Kelley; Joyner; Davis; Baccanari
Journal of Medicinal Chemistry, 1995 , vol. 38, # 19 p. 3850 - 3856