甲苯-4-磺酸氧杂环丁-3-基酯合成路线 (共 2 条)
反应条件
triethylamine in water T=20°C; 18 h;
参考文献
MERCK SHARP and DOHME CORP.; WU, Wen-Lian; BURNETT, Duane, A.; GREENLEE, William, J.
Patent: WO2012/138678 A1, 2012 ;
Location in patent: Page/Page column 33 ;
反应条件
potassium iodide in 1,2-bis-(2-hydroxyethoxy)-ethane P=10 Torr; Heating;
参考文献
Duncton, Matthew A. J.; Estiarte, M. Angels; Tan, Darlene; Kaub, Carl; O'Mahony, Donogh J. R.; Johnson, Russell J.; Cox, Matthew; Edwards, William T.; Wan, Min; Kincaid, John; Kelly, Michael G.
Organic Letters, 2008 , vol. 10, # 15 p. 3259 - 3262