反应条件
1: 1.) Mg, 2.) dilithium tetrachlorocopper(II) / 1.) THF, reflux, 2 h, 2.) a) THF, reflux, 2 h, b) THF, RT, 16 h
2: 94 percent / BBr3 / CH2Cl2 / 3 h / Ambient temperature
View Scheme
参考文献
Wissner; Sum; Schaub; Kohler; Goldstein
Journal of Medicinal Chemistry, 1984 , vol. 27, # 9 p. 1174 - 1181
