1: S-(3-nitrophenyl) dimethylthiocarbamate With potassium hydroxide in methanol; water 2 h; Heating / reflux; 2: dimethyl sulfate in methanol; water T=20°C; 16 h;
Hay, Michael P.; Gamage, Swarna A.; Kovacs, Mary S.; Pruijn, Frederik B.; Anderson, Robert F.; Patterson, Adam V.; Wilson, William R.; Brown, J. Martin; Denny, William A.
Journal of Medicinal Chemistry, 2003 , vol. 46, # 1 p. 169 - 182