1: With (2S,3S)-2-(tert-butoxycarbonylamino)-3-methylpentanoic acid; oxygen; palladium diacetate; potassium hydrogencarbonate in 1,1-dimethylpropan-1-ol T=90°C; P=760.051 Torr; 2: With hydrogenchloride in 1,1-dimethylpropan-1-ol; water T=20°C; pH=1;
参考文献
Baxter, Ryan D.; Sale, David; Engle, Keary M.; Yu, Jin-Quan; Blackmond, Donna G.
Journal of the American Chemical Society, 2012 , vol. 134, # 10 p. 4600 - 4606