1: With lithium aluminium tetrahydride in tetrahydrofuran
T=0 - 20°C; Heating / reflux;
2: With sodium hydroxide in tetrahydrofuran; water
T=0 - 20°C; 1 h;
参考文献
SGX Pharmaceuticals, Inc.
Patent: US2007/173488 A1, 2007 ;
Location in patent: Page/Page column 52 ;