反应条件
1.1: (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride / tetrahydrofuran / 1.5 h / 85 °C / |Inert atmosphere 2.1: water; lithium hydroxide hydrate / tetrahydrofuran / 20 °C 2.2: 5 h / 50 °C View Scheme
参考文献
BOEHRINGER INGELHEIM INTERNATIONAL GMBH; HEIMANN, Annekatrin; DAHMANN, Georg; GRUNDL, Marc; MUELLER, Stephan Georg; WELLENZOHN, Bernd
Patent: WO2013/87805 A1, 2013 ;