H-顺式-4-氟-脯氨酸合成路线 (共 12 条)
反应条件
triethylamine in methanol Yield given;
参考文献
Tetrahedron Letters, , vol. 39, # 10 p. 1169 - 1172
反应条件
1: With hydrogenchloride in ethanol
T=20 - 55°C; 62 h;
2: With ammonia in methanol; water
T=20°C; 36 h;
参考文献
NOVARTIS AG
Patent: US2011/3786 A1, 2011 ;
Location in patent: Page/Page column 20-21 ;
US 20110003786 A1