反应条件
1: 66 percent / Et3N / butan-1-ol / 22 h / Heating
2: 63 percent / diethyl ether / 1.) 35-40 deg C, 4 h, 2.) ca. 20 deg C, 16 h
View Scheme
参考文献
Lukevits, E.; Veveris, M. M.; Atare, Z. A.; Segal, I. D.; Khokhlova, L. N.; Kimenis, A. A.
Pharmaceutical Chemistry Journal, 1982 , vol. 16, # 10 p. 764 - 768
Khimiko-Farmatsevticheskii Zhurnal, 1982 , vol. 16, # 10 p. 1204 - 1209