反应条件
1: With diphenyl-phosphinic acid; triethylamine in N,N-dimethyl-formamide
T=20°C; 3 h;
2: With water in N,N-dimethyl-formamide
1 h; Heating;
参考文献
Jia, Zhaozhong J.; Wu, Yanhong; Huang, Wenrong; Zhang, Penglie; Song, Yonghong; Woolfrey, John; Sinha, Uma; Arfsten, Ann E.; Edwards, Susan T.; Hutchaleelaha, Athiwat; Hollennbach, Stanley J.; Lambing, Joseph L.; Scarborough, Robert M.; Zhu, Bing-Yan
Bioorganic and Medicinal Chemistry Letters, 2004 , vol. 14, # 5 p. 1229 - 1234