4-[(4-甲基苯基)磺酰基]苯胺合成路线 （共 16 条）
反应条件
hydrogen; Raney Ni (W2) in methanol T=45°C; P=3000.2 Torr; 6 h;
参考文献
Kansy, M; Seydel, JK; Wiese, M; Haller, R
European Journal of Medicinal Chemistry, 1992 , vol. 27, # 3 p. 237 - 244
反应条件
CyPF-tBu; palladium diacetate; lithium hexamethyldisilazane in ethylene glycol dimethyl ether T=90°C; Inert atmosphere;
参考文献
Fernandez-Rodriguez, Manuel A.; Hartwig, John F.
Journal of Organic Chemistry, 2009 , vol. 74, # 4 p. 1664 - 1672
反应条件
potassium hydroxide in poly(ethylene glycol)-600 T=100°C; 2 h;
参考文献
Duan, Zhongyu; Ranjit, Sadananda; Liu, Xiaogang
Organic Letters, 2010 , vol. 12, # 10 p. 2430 - 2433
反应条件
potassium carbonate in N,N-dimethyl-formamide T=120°C; 0.0833333 h; microwave irradiation;
参考文献
Advanced Synthesis and Catalysis, , vol. 349, # 17-18 p. 2690 - 2696
反应条件
copper(l) iodide; 8-Hydroxyquinoline 1-oxide; caesium carbonate in dimethyl sulfoxide T=80°C; 24 h; Inert atmosphere; chemoselective reaction;
参考文献
Su, Kun; Qiu, Yatao; Yao, Yiwu; Zhang, Dayong; Jiang, Sheng
Synlett, 2012 , vol. 23, # 19 p. 2853 - 2857
反应条件
1.1: K2CO3; Cu / dimethylformamide / 0.25 h 1.2: 61 percent / dimethylformamide / 150 °C 2.1: 73 percent / SnCl2*2H2O / ethanol / 70 °C View Scheme
参考文献
Farmaco, , vol. 59, # 6 p. 443 - 450
反应条件
iron(III) trifluoride; iodine in acetonitrile T=80°C; 36 h; Inert atmosphere; regioselective reaction;
参考文献
Fang, Xiao-Li; Tang, Ri-Yuan; Zhang, Xing-Guo; Li, Jin-Heng
Synthesis, 2011 , # 7 p. 1099 - 1105
反应条件
tetrabutyl ammonium fluoride; palladium diacetate; NAF in water T=150°C; 0.333333 h; Microwave irradiation;
参考文献
Synlett, , # 18 p. 2733 - 2736
反应条件
1: dimethylformamide / 120 °C 2: SnCl2 / ethanol / Heating View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 14, # 4 p. 1053 - 1056
反应条件
copper(I) sulphide; iron; potassium carbonate; dimethyl sulfoxide T=110°C; 24 h; Inert atmosphere; chemoselective reaction;
参考文献
Wang, Huifeng; Jiang, Linlin; Chen, Tao; Li, Yarning
European Journal of Organic Chemistry, 2010 , # 12 p. 2324 - 2329
