8-甲氧基-1,3,4,5-四氢-苯并[B]氮杂革-2-酮合成路线 （共 6 条）
反应条件
sodium azide; PPA T=55°C;
参考文献
CEPHALON, INC.; PHARMACOPEIA DRUG DISCOVERY, INC.
Patent: WO2008/51547 A1, 2008 ;
Location in patent: Page/Page column 361 ;
WO 2008/051547 A1
反应条件
PPA T=115°C; Beckman rearrangement; 0.0833333 h;
参考文献
Antex Pharma Inc.
Patent: US6514965 B1, 2003 ;
反应条件
hydrogenchloride; sodium azide in water T=0 - 50°C; Schmidt reaction;
参考文献
Crosby, Ian T.; Shin, James K.; Capuano, Ben
Australian Journal of Chemistry, 2010 , vol. 63, # 2 p. 211 - 226
参考文献
BYK Gulden Lomberg Chemische Fabrik GmbH
Patent: US4322439 A1, 1982 ;
参考文献
Ciba-Geigy Corporation
Patent: US4575503 A1, 1986 ;
Title/Abstract Full Text Show Details
Ciba-Geigy Corporation
Patent: US4473575 A1, 1984 ;
反应条件
boron tribromide in 4-(dicyanomethylene)-2-methyl-6-(4-dimethylaminostyryl)-4H-pyran
参考文献
Antex Pharma Inc.
Patent: US6514965 B1, 2003 ;
