8-甲氧基-2,3,4,5-四氢苯并氮杂卓-1-酮合成路线 （共 4 条）
反应条件
hydrogenchloride; sodium azide T=20°C; 2 h;
参考文献
Ueno, Hiroshi; Yokota, Katsuyuki; Hoshi, Jun-Ichi; Yasue, Katsutaka; Hayashi, Mikio; Hase, Yasunori; Uchida, Itsuo; Aisaka, Kazuo; Katoh, Susumu; Cho, Hidetsura
Journal of Medicinal Chemistry, 2005 , vol. 48, # 10 p. 3586 - 3604
反应条件
hydrogenchloride; sodium azide in water T=0 - 50°C; Schmidt reaction;
参考文献
Crosby, Ian T.; Shin, James K.; Capuano, Ben
Australian Journal of Chemistry, 2010 , vol. 63, # 2 p. 211 - 226
反应条件
trichloroacetic acid
参考文献
Genentech, Inc.
Patent: US5250679 A1, 1993 ;
反应条件
lithium aluminium tetrahydride in tetrahydrofuran; 1,4-dioxane 20 h; Heating;
参考文献
MERCK and CO., INC.
Patent: WO2008/54605 A2, 2008 ;
Location in patent: Page/Page column 68 ;
WO 2008/054605 A2
