6-溴-8-甲基-咪唑并[1,2-a]吡啶合成路线 (共 3 条)
反应条件
in ethanol 4 h; Heating;
参考文献
Gueiffier; Mavel; Lhassani; Elhakmaoui; Snoeck; Andrei; Chavignon; Teulade; Witvrouw; Balzarini; De Clercq; Chapat
Journal of Medicinal Chemistry, 1998 , vol. 41, # 25 p. 5108 - 5112
反应条件
in ethanol 24 h; Reflux;
参考文献
Veron, Jean-Baptiste; Allouchi, Hassan; Enguehard-Gueiffier, Cecile; Snoeck, Robert; Andrei, Graciela; De Clercq, Erik; Gueiffier, Alain
Bioorganic and Medicinal Chemistry, 2008 , vol. 16, # 21 p. 9536 - 9545
参考文献
Eisai Co., Ltd.
Patent: EP1382603 A1, 2004 ;
Location in patent: Page 135 ;