反应条件
1: 2,4-dibromo-1,3-thiazole With n-butyllithium in tetrahydrofuran T=-78°C; 0.5 h; 2: 4-acetylmorpholine in tetrahydrofuran T=-78°C; 2 h; Further stages.;
参考文献
Gebauer, Julian; Arseniyadis, Stellios; Cossy, Janine
Organic Letters, 2007 , vol. 9, # 17 p. 3425 - 3427