1: With sodium azide in 1-methyl-pyrrolidin-2-one; water T=70°C; 3 h; 2: With sodium tetrahydroborate in 1-methyl-pyrrolidin-2-one; water T=50 - 70°C; 3 h;
参考文献
Torisawa, Yasuhiro; Nishi, Takao; Minamikawa, Jun-ichi
Bioorganic and Medicinal Chemistry, 2002 , vol. 10, # 8 p. 2583 - 2587