N-叔-丁氧羰基-4-氯-2-三氟乙酰基苯胺合成路线 (共 1 条)
反应条件
1: cyclopropyl acetylene With n-butyllithium in tetrahydrofuran; hexane T=0°C; 2: C13H13ClF3NO3 in tetrahydrofuran; hexane T=-70 - 65°C; 2.5 h; Heating / reflux;
参考文献
Pierce, Michael Ernest; Radesca, Lilian Alicia
Patent: US6348616 B1, 2002 ;
Location in patent: Page column 24 ;