反应条件
potassium carbonate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in 1,4-dioxane; water
T=80°C; 15 h;
参考文献
MERCK SHARP and DOHME CORP.; MERCK CANADA INC.; DESCHENES, Denis; ALTMAN, Michael, D.; ELLIS, John Michael; FISCHER, Christian; HAIDLE, Andrew, M.; KATTAR, Solomon, D.; NORTHRUP, Alan, B.; SCHELL, Adam, J.; SMITH, Graham, F.; TAOKA, Brandon, M.; BIENSTOCK, Corey; DI FRANCESCO, Maria Emilia; DONOFRIO, Anthony; PETERSON, Scott; SPENCER, Kerrie, B.; JEWELL, James Patrick; ALI, Amjad; BENNETT, David Jonathan; DANG, Qun; WAI, John
Patent: WO2012/154518 A1, 2012 ;
Location in patent: Page/Page column 44 ;
WO 2012/154518 A1