反应条件
dicyclohexyl-carbodiimide 1.) THF, -15 deg C, 5 min, 2.) THF, a) -10 deg C, 30 min, b) 0 deg C, 4 h; Yield given. Multistep reaction;
参考文献
Qasmi, Driss; De Rosny, Eve; Rene, Loic; Badet, Bernard; Vergely, Isabelle; Boggetto, Nicole; Reboud-Ravaux, Michele
Bioorganic and Medicinal Chemistry, 1997 , vol. 5, # 4 p. 707 - 714