N-Boc-六氢-1H-氮杂卓-4-酮合成路线

参考文献

MORPHOCHEM AKTIENGESELLSCHAFT FUeR KOMBINATORISCHE CHEMIE
Patent: WO2004/35569 A2, 2004 ;
Location in patent: Page/Page column 58 ;

24424-99-5二碳酸二叔丁酯+

1208-75-91-苄基六氢氮杂卓-4-酮

188975-88-4N-Boc-六氢-1H-氮杂卓-4-酮

参考文献

JANSSEN RandD IRELAND; GUILLEMONT, Jerôme Emile Georges; LANÇOIS, David Francis Alain; MOTTE, Magali Madeleine Simone; BALEMANS, Wendy Mia Albert; KOUL, Anil
Patent: WO2014/23815 A1, 2014 ;
Location in patent: Page/Page column 37 ;

478832-21-24-羟基氮杂环庚烷-1-羧酸叔丁酯

188975-88-4N-Boc-六氢-1H-氮杂卓-4-酮

参考文献

Sumitomo Pharmaceuticals Company, Limited
Patent: EP1500643 A1, 2005 ;
Location in patent: Page 48 ;
EP 1500643 A1

24424-99-5二碳酸二叔丁酯+

50492-22-34-氮杂卓酮盐酸盐

188975-88-4N-Boc-六氢-1H-氮杂卓-4-酮

参考文献

SMITHKLINE BEECHAM CORPORATION
Patent: WO2007/30366 A1, 2007 ;
Location in patent: Page/Page column 130 ;

105416-56-6氮杂环庚-4-酮+

24424-99-5二碳酸二叔丁酯

188975-88-4N-Boc-六氢-1H-氮杂卓-4-酮

参考文献

ELI LILLY AND COMPANY
Patent: WO2009/12125 A1, 2009 ;
Location in patent: Page/Page column 29-30 ;

24424-99-5二碳酸二叔丁酯+

1208-76-01-苄基-4-氧代氮杂烷盐酸盐

188975-88-4N-Boc-六氢-1H-氮杂卓-4-酮

参考文献

JANSSEN RandD IRELAND; GUILLEMONT, Jerôme Emile Georges; LANÇOIS, David Francis Alain; MOTTE, Magali Madeleine Simone; BALEMANS, Wendy Mia Albert; KOUL, Anil
Patent: WO2014/23815 A1, 2014 ;
Location in patent: Page/Page column 43 ;

24424-99-5二碳酸二叔丁酯

188975-88-4N-Boc-六氢-1H-氮杂卓-4-酮

参考文献

Millennium Pharmaceuticals, Inc.
Patent: US2002/169155 A1, 2002 ;
US 20020169155 A1

623-73-4重氮乙酸乙酯+

79099-07-3N-叔丁氧羰基-4-哌啶酮

188975-88-4N-Boc-六氢-1H-氮杂卓-4-酮

参考文献

WO2008/65500 A2, ;

Page/Page column 51; 52 ;
WO 2008/065500 A2

79099-07-3N-叔丁氧羰基-4-哌啶酮

188975-88-4N-Boc-六氢-1H-氮杂卓-4-酮

参考文献