3-氨基-6-碘哒嗪合成路线

参考文献

F. HOFFMANN-LA ROCHE AG; HOFFMANN-LA ROCHE INC.; FLOHR, Alexander; GROEBKE ZBINDEN, Katrin; KOERNER, Matthias; LERNER, Christian
Patent: WO2013/178569 A1, 2013 ;
Location in patent: Page/Page column 58-59 ;

1679-18-14-氯苯硼酸+

187973-60-03-氨基-6-碘哒嗪

58059-47-53-氨基-6-(4-氯苯基)哒嗪

参考文献

Maes, Bert U. W.; Lemiere, Guy L. F.; Dommisse, Roger; Augustyns, Koen; Haemers, Achiel
Tetrahedron, 2000 , vol. 56, # 12 p. 1777 - 1781

5720-07-04-甲氧基苯硼酸+

187973-60-03-氨基-6-碘哒嗪

4776-87-83-氨基-6-(4-甲氧基苯基)哒嗪

参考文献

Maes, Bert U. W.; Lemiere, Guy L. F.; Dommisse, Roger; Augustyns, Koen; Haemers, Achiel
Tetrahedron, 2000 , vol. 56, # 12 p. 1777 - 1781

1005786-10-6

参考文献

TAKEDA PHARMACEUTICAL COMPANY LIMITED
Patent: US2009/137595 A1, 2009 ;

40235-68-51-乙酰氧基-3-氯丙酮+

144-55-8碳酸氢钠+

187973-60-03-氨基-6-碘哒嗪

1005788-25-9

参考文献

US2009/137595 A1, ;

6092-47-3N-氯乙酰氨基甲酸+

187973-60-03-氨基-6-碘哒嗪

1005785-69-2

参考文献

Bioorganic and Medicinal Chemistry, , vol. 21, # 8 p. 2333 - 2345

1005785-69-2

参考文献

US2009/137595 A1, ;

187973-60-03-氨基-6-碘哒嗪+

98-80-6苯硼酸

14966-91-76-苯基-3-氨基哒嗪

参考文献

Maes, Bert U. W.; Lemiere, Guy L. F.; Dommisse, Roger; Augustyns, Koen; Haemers, Achiel
Tetrahedron, 2000 , vol. 56, # 12 p. 1777 - 1781