3-(2-乙氧基-2-氧代乙氧基)异烟酸乙酯合成路线 (共 11 条)
反应条件
1: sodium hydride / tetrahydrofuran; mineral oil / 16 h / 0 - 20 °C / |Inert atmosphere
2: pyridine / dichloromethane / 16 h / 0 - 20 °C
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参考文献
GENENTECH,INC.; FORMA TM, LLC; YUEN, Po-Wai; BAIR, Kenneth, W.; BAUMEISTER, Timm, R.; DRAGOVICH, Peter; LIU, Xiongcai; PATEL, Snahel; ZAK, Mark; ZHAO, Guiling; ZHANG, Yamin; ZHENG, Xiaozhang
Patent: WO2013/127269 A1, 2013 ;