反应条件
1: 1.) NaH / 1.) THF, 0 deg C, 0.5 h, 2.) THF, 15 min
2: 98 percent / H2 / Pd/C / methanol / 258.6 Torr
View Scheme
参考文献
Chandrakumar; Yonan; Stapelfeld; Savage; Rorbacher; Contreras; Hammond
Journal of Medicinal Chemistry, 1992 , vol. 35, # 2 p. 223 - 233