1-羟基-3H-吲哚-2-酮合成路线 （共 19 条）
反应条件
water; hydrogen bromide T=100°C;
参考文献
Wright; Collins
Journal of the American Chemical Society, 1956 , vol. 78, p. 221,222
参考文献
Wright; Collins
Journal of the American Chemical Society, 1956 , vol. 78, p. 221,222
反应条件
diethylamino-sulfur trifluoride in dichloromethane T=0°C; 0.0833333 h;
参考文献
Kikugawa, Yasuo; Matsumoto, Kazuhiro; Mitsui, Kimiyo; Sakamoto, Takeshi
Journal of the Chemical Society, Chemical Communications, 1992 , # 12 p. 921 - 922
反应条件
1: 95 percent / PPh3, diethyl diazocarbonate / CHCl3 / 1 h 2: 88.2 percent / DIBAL / toluene; tetrahydrofuran / 1 h / -78 °C 3: (n-Bu)4NF / tetrahydrofuran / 2 h / Ambient temperature View Scheme
参考文献
Henmi, Toshiyuki; Sakamoto, Takeshi; Kikugawa, Yasuo
Heterocycles, 1997 , vol. 44, # 1 p. 157 - 163
反应条件
1: water; NaOH-solution 2: hydrochloric acid; water / 100 °C View Scheme
参考文献
Wright; Collins
Journal of the American Chemical Society, 1956 , vol. 78, p. 221,222
参考文献
Bourque, Jennifer R.; Burley, Rodney K.M.; Bearne, Stephen L.
Bioorganic and Medicinal Chemistry Letters, 2007 , vol. 17, # 1 p. 105 - 108
反应条件
ammonium chloride; zinc in methanol; water
T=20°C; 3 h;
参考文献
Somei; Yamada; Kurauchi; Nagahama; Hasegawa; Teranishi; Sato; Kaneko
Chemical and Pharmaceutical Bulletin, 2001 , vol. 49, # 1 p. 87 - 96
反应条件
sodium hypophosphite; palladium on activated charcoal in tetrahydrofuran
T=20°C;
参考文献
Yoneyama, Hiroki; Shimoda, Ayako; Araki, Lisa; Hatano, Kouta; Sakamoto, Yasuhiko; Kurihara, Takushi; Yamatodani, Atsushi; Harusawa, Shinya
Journal of Organic Chemistry, 2008 , vol. 73, # 6 p. 2096 - 2104
反应条件
3,3-dimethyldioxirane in acetone
T=0°C;
参考文献
Neset, Siren Marcussen; Benneche, Tore; Undheim, Kjell
Acta Chemica Scandinavica, 1993 , vol. 47, # 11 p. 1141 - 1143
反应条件
palladium diacetate; triethylammonium formate; triphenylphosphine in ethanol; water
0.166667 h; Heating;
参考文献
Kikugawa, Yasuo; Shimada, Masahiro; Matsumoto, Kazuhiro
Heterocycles, 1994 , vol. 37, # 1 p. 293 - 302
