1-Boc-2-羟基甲基-氮杂丁烷合成路线 (共 2 条)
反应条件
hydrogen; palladium dihydroxide in ethanol
参考文献
Evans, Gary B.; Furneaux, Richard H.; Greatrex, Ben; Murkin, Andrew S.; Schramm, Vern L.; Tyler, Peter C.
Journal of Medicinal Chemistry, 2008 , vol. 51, # 4 p. 948 - 956
反应条件
1: With sodium tetrahydroborate in tetrahydrofuran Heating / reflux; 2: With methanol in tetrahydrofuran 1.5 h; Heating / reflux;
参考文献
US2003/229226 A1, ;
Page 19 ;