6-氯吲哚合成路线

参考文献

Oelke, Alexander J.; Antonietti, Francesca; Bertone, Leonardo; Cranwell, Philippa B.; France, David J.; Goss, Rebecca J. M.; Hofmann, Tatjana; Knauer, Stephan; Moss, Steven J.; Skelton, Paul C.; Turner, Richard M.; Wuitschik, Georg; Ley, Steven V.
Chemistry - A European Journal, 2011 , vol. 17, # 15 p. 4183 - 4194

17422-33-26-氯吲哚

50517-12-9氯克胺

参考文献

POLIFARMA S.p.A.
Patent: EP421946 A2, 1991 ;

参考文献

Hall, Adrian; Billinton, Andy; Brown, Susan H.; Chowdhury, Anita; Giblin, Gerard M.P.; Goldsmith, Paul; Hurst, David N.; Naylor, Alan; Patel, Sadhana; Scoccitti, Tiziana; Theobald, Pamela J.
Bioorganic and Medicinal Chemistry Letters, 2008 , vol. 18, # 8 p. 2684 - 2690

17422-33-26-氯吲哚+

302-84-1丝氨酸+

108-24-7乙酸酐

50517-10-7N-乙酰基6-氯色氨酸

参考文献

Bioorganic and Medicinal Chemistry, , vol. 21, # 5 p. 1159 - 1165

17422-33-26-氯吲哚+

56-45-1L-丝氨酸+

108-24-7乙酸酐

50517-10-7N-乙酰基6-氯色氨酸

参考文献

Tetrahedron Letters, , vol. 49, # 17 p. 2795 - 2798

17422-33-26-氯吲哚+

40064-34-44,4-哌啶二醇盐酸盐

180160-69-4+

180160-77-46-氯-3-(1,2,3,6-四氢吡啶-4-基)-1H-吲哚

参考文献

Eli Lilly and Company
Patent: US5627196 A1, 1997 ;

Title/Abstract Full Text Show Details
Eli Lilly Company
Patent: US5789402 A1, 1998 ;
US 5789402 A
Title/Abstract Full Text Show Details
Eli Lilly and Company
Patent: US5614523 A1, 1997 ;
US 5614523 A

17422-33-26-氯吲哚+

40064-34-44,4-哌啶二醇盐酸盐

180160-77-46-氯-3-(1,2,3,6-四氢吡啶-4-基)-1H-吲哚

参考文献

Eli Lilly and Company
Patent: US5846982 A1, 1998 ;
US 5846982 A

17422-33-26-氯吲哚+

107-14-2氯乙腈

1912-44-36-氯吲哚-3-乙酸

参考文献

Fox; Bullock
Journal of the American Chemical Society, 1951 , vol. 73, p. 2756,2758

17422-33-26-氯吲哚

1912-44-36-氯吲哚-3-乙酸

参考文献

Lozano, Oscar; Blessley, George; Martinez Del Campo, Teresa; Thompson, Amber L.; Giuffredi, Guy T.; Bettati, Michela; Walker, Matthew; Borman, Richard; Gouverneur, Veronique
Angewandte Chemie - International Edition, 2011 , vol. 50, # 35 p. 8105 - 8109

17422-33-26-氯吲哚

52537-00-56-氯-2,3-二氢-1H-吲哚

参考文献

ELI LILLY AND COMPANY
Patent: WO2003/76398 A2, 2003 ;
Location in patent: Page/Page column 41 ;
WO 03/076398 A2