4-氨基-N-[(2R, 3S)-3-氨基-2-羟基-4-苯丁基]-N-异丁基苯磺酰胺合成路线

159005-59-1

169280-56-24-氨基-N-[(2R, 3S)-3-氨基-2-羟基-4-苯丁基]-N-异丁基苯磺酰胺

参考文献

Ajinomoto Co., Inc.
Patent: EP1466896 A1, 2004 ;
Location in patent: Page 12-13 ;

143224-62-8+

98-74-8对硝基苯磺酰氯

169280-56-24-氨基-N-[(2R, 3S)-3-氨基-2-羟基-4-苯丁基]-N-异丁基苯磺酰胺

参考文献

Ajinomoto Co., Inc.
Patent: EP1466896 A1, 2004 ;
Location in patent: Page 14-15 ;

191226-98-9[(1S,2R)-1-苄基-2-羟基-3-[异丁基[(4-硝基苯基)磺酰]氨基]丙基]氨基甲酸叔丁酯

169280-56-24-氨基-N-[(2R, 3S)-3-氨基-2-羟基-4-苯丁基]-N-异丁基苯磺酰胺

参考文献

MATRIX LABORATORIES LIMITED; VELLANKI, Siva Rama Prasad; SAHU, Arabinda; KATUKURI, Aravind Kumar; VANAMA, Vikram; KOTHARI, Satishbabu; PONNEKANTI, Venkata Suryanarayana; DATTA, Debashish
Patent: WO2011/48604 A2, 2011 ;
Location in patent: Page/Page column 19 ;

183004-94-6[(1S,2R)-1-苄基-2-羟基-3-[异丁基-[(4-氨基苯基)磺酰基]氨基] 丙基]氨基甲酸叔丁酯

169280-56-24-氨基-N-[(2R, 3S)-3-氨基-2-羟基-4-苯丁基]-N-异丁基苯磺酰胺

参考文献

Yeung, Clinton M.; Klein, Larry L.; Flentge, Charles A.; Randolph, John T.; Zhao, Chen; Sun, MingHua; Dekhtyar, Tatyana; Stoll, Vincent S.; Kempf, Dale J.
Bioorganic and Medicinal Chemistry Letters, 2005 , vol. 15, # 9 p. 2275 - 2278

244641-42-7

169280-56-24-氨基-N-[(2R, 3S)-3-氨基-2-羟基-4-苯丁基]-N-异丁基苯磺酰胺

参考文献

Surleraux, Dominique L. N. G.; Tahri, Abdellah; Verschueren, Wim G.; Pille, Geert M. E.; De Kock, Herman A.; Jonckers, Tim H. M.; Peeters, Anik; De Meyer, Sandra; Azijn, Hilde; Pauwels, Rudi; De Bethune, Marie-Pierre; King, Nancy M.; Prabu-Jeyabalan, Moses; Schiffer, Celia A.; Wigerinck, Piet B. T. P.
Journal of Medicinal Chemistry, 2005 , vol. 48, # 6 p. 1813 - 1822

251105-80-3

169280-56-24-氨基-N-[(2R, 3S)-3-氨基-2-羟基-4-苯丁基]-N-异丁基苯磺酰胺

参考文献

RANBAXY LABORATORIES LIMITED; JAYACHANDRA, Suresh, Babu; YOGESH, Ruchika; NAGDA, Devendra, Prakash; KHANDURI, Chandra, Has
Patent: WO2013/11485 A1, 2013 ;
Location in patent: Page/Page column 23 ;
WO 2013/011485 A1

1415750-61-6

169280-56-24-氨基-N-[(2R, 3S)-3-氨基-2-羟基-4-苯丁基]-N-异丁基苯磺酰胺

参考文献

WO2005/63770 A1, ;

Page/Page column 27 ;
WO 2005/063770 A1

160230-47-7

169280-56-24-氨基-N-[(2R, 3S)-3-氨基-2-羟基-4-苯丁基]-N-异丁基苯磺酰胺

参考文献

RANBAXY LABORATORIES LIMITED; JAYACHANDRA, Suresh, Babu; YOGESH, Ruchika; NAGDA, Devendra, Prakash; KHANDURI, Chandra, Has
Patent: WO2013/11485 A1, 2013 ;
Location in patent: Page/Page column 33 ;
WO 2013/011485 A1

98760-08-8(1S)-1-(2R)-环氧乙基-2-苯乙基氨基甲酸叔丁酯

169280-56-24-氨基-N-[(2R, 3S)-3-氨基-2-羟基-4-苯丁基]-N-异丁基苯磺酰胺

参考文献

Bioorganic and Medicinal Chemistry, , vol. 14, # 19 p. 6695 - 6712

160232-08-6[(1S,2R)-2-羟基-3-[(2-甲基丙基)氨基]-1-(苯基甲基)丙基]-1,1,-二甲基乙酯

169280-56-24-氨基-N-[(2R, 3S)-3-氨基-2-羟基-4-苯丁基]-N-异丁基苯磺酰胺

参考文献

Bioorganic and Medicinal Chemistry, , vol. 14, # 19 p. 6695 - 6712