反应条件
1.1: sodium hydride / mineral oil; tetrahydrofuran / 1 h / 0 - 20 °C 1.2: 1 h / 0 °C 2.1: sodium hydrogencarbonate / 1,4-dioxane / 3 h / 20 - 80 °C 3.1: NH2NH2•xH2O / ethanol / 2 h / 20 - 90 °C View Scheme
参考文献
CENTAURUS BIOPHARMA CO., LTD.; HAN, Yongxin; YU, Rong; WANG, Zanping; LIANG, Zhi; HU, Quan; ZHU, Li; HU, Yuandong; SUN, Yinghui; ZHAO, Na; PENG, Yong; ZHAI, Xiaofeng; LUO, Hong; XIAO, Dengming
Patent: WO2014/82598 A1, 2014 ;