反应条件
sodium methylate; acetic acid 1.) MeOH, reflux, 4 h, 2.) MeOH, reflux, 18 h; Multistep reaction;
参考文献
Patt, William C.; Cheng, Xue-Min; Repine, Joseph T.; Lee, Chet; Reisdorph, Bill R.; Massa, Mark A.; Doherty, Annette M.; Welch, Kathleen M.; Bryant, John W.; Flynn, Michael A.; Walker, Donnelle M.; Schroeder, Richard L.; Haleen, Stephen J.; Keiser, Joan A.
Journal of Medicinal Chemistry, 1999 , vol. 42, # 12 p. 2162 - 2168