反应条件
1: 1.) Mg / 1.) THF, 0 deg C, 2 h, 2.) THF, overnight
2: 88 percent / benzene / 18 h / Heating
View Scheme
参考文献
Vaccaro, Wayne; Amore, Cindy; Berger, Joel; Burrier, Robert; Clader, John; Davis, Harry; Domalski, Martin; Fevig, Tom; Salisbury, Brian; Sher, Rosy
Journal of Medicinal Chemistry, 1996 , vol. 39, # 8 p. 1704 - 1719