反应条件
1: 100 percent / 1-methyl-pyrrolidin-2-one / 0.17 h / 160 °C / microwave irradiation
2: 75 percent / K2CO3; (1R,2R)-1,2-cyclohexanebis(methylamine) / CuI / 1-methyl-pyrrolidin-2-one / 0.17 h / 160 °C / microwave irradiation
View Scheme
参考文献
Pabba, Chittari; Wang, Hong-Jun; Mulligan, Susan R.; Chen, Zhen-Jia; Stark, Todd M.; Gregg, Brian T.
Tetrahedron Letters, 2005 , vol. 46, # 44 p. 7553 - 7557