反应条件
1: 1.) Et3N, ethyl chloroformate, 2.) NH3 gas / 1.) THF, 30 min, 2.) THF, 3 h 2: 1.) NaH / 1.) DMF, 1 h ,2.) DMF, 4 h View Scheme
参考文献
Dillard, Robert D.; Bach, Nicholas J.; Draheim, Susan E.; Berry, Dennis R.; Carlson, Donald G.; Chirgadze, Nickolay Y.; Clawson, David K.; Hartley, Lawrence W.; Johnson, Lea M.; Jones, Noel D.; McKinney, Emma R.; Mihelich, Edward D.; Olkowski, Jennifer L.; Schevitz, Richard W.; Smith, Amy C.; Snyder, David W.; Sommers, Cynthia D.; Wery, Jean-Pierre
Journal of Medicinal Chemistry, 1996 , vol. 39, # 26 p. 5119 - 5136
