反应条件
1: 1.) acetic anhydride / 1.) 50 deg C - 60 deg C, 2 h, 2.) THF, RT, 18 h 2: 1.) borane dimethyl sulfide complex, 2.) HCl / 1.) THF, reflux, 18 h, 2.) THF, CH3OH, reflux, 1.5 h View Scheme
参考文献
Romero; Morge; Biles; Berrios-Pena; May; Palmer; Johnson; Smith; Busso; Tan; Voorman; Reusser; Althaus; Downey; So; Resnick; Tarpley; Aristoff
Journal of Medicinal Chemistry, 1994 , vol. 37, # 7 p. 999 - 1014
