反应条件
1: 3-cyclopropyl-1-(2-fluorophenyl)-3-oxopropyl methanesulfonate; 2-oxo-2,4,5,6,7a-hexahydrothieno[3,2-c]pyridine hydrochloride With tetraethylammonium bromide; N-ethyl-N,N-diisopropylamine in acetonitrile T=20°C; 1.5 h; 2: acetic anhydride With N-ethyl-N,N-diisopropylamine; 4-(N,N-dimethlyamino)pyridine in acetonitrile T=20°C; 2 h;