反应条件
1: 2-amino-benzonitrile With sodium methylate in 1,4-dioxane Deprotonation; 2: hydrogen cyanide in 1,4-dioxane Cycloaddition; 16 h; Heating; Further stages.;
参考文献
Van Muijlwijk-Koezen, Jacqueline E.; Timmerman, Henk; Van Der Goot, Henk; Menge, Wiro M. P. B.; Von Drabbe Kuenzel, Jacobien Frijtag; De Groote, Miriam; Ijzerman, Adriaan P.
Journal of Medicinal Chemistry, 2000 , vol. 43, # 11 p. 2227 - 2238