5-氯-3,4-二氢喹噁啉-2(1h)-酮合成路线 (共 1 条)
反应条件
1: 3percent aq. H2O2; aq. NaOH / 1 h / Heating
2: 70 percent / POCl3 / 1 h / Heating
View Scheme
参考文献
Hazeldine; Polin; Kushner; Paluch; White; Edelstein; Palomino; Corbett; Horwitz
Journal of Medicinal Chemistry, 2001 , vol. 44, # 11 p. 1758 - 1776