1-Boc-4-烯丙基-4-哌啶甲酸乙酯合成路线

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参考文献

Pineiro, Jose Luis Castro; Dinnell, Kevin; Elliott, Jason Matthew; Hollingworth, Gregory John; Shaw, Duncan Edward; Swain, Christopher John; Yang, Lihu
Patent: US2003/225059 A1, 2003 ;
Location in patent: Page 27 ;

556-56-9丙烯酰碘+

142851-03-4N-Boc-4-哌啶甲酸乙酯

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146603-99-81-Boc-4-烯丙基-4-哌啶甲酸乙酯

参考文献

SANOFI; GAO, Zhongli; HALL, Daniel; STEFANY, David
Patent: WO2011/143148 A1, 2011 ;
Location in patent: Page/Page column 25-26 ;
WO 2011/143148 A1

5162-44-74-溴-1-丁烯+

142851-03-4N-Boc-4-哌啶甲酸乙酯

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146603-99-81-Boc-4-烯丙基-4-哌啶甲酸乙酯

参考文献

SANOFI; GAO, Zhongli
Patent: WO2011/143150 A1, 2011 ;
Location in patent: Page/Page column 33-34 ;
WO 2011/143150 A1

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146603-99-81-Boc-4-烯丙基-4-哌啶甲酸乙酯

参考文献

US6562828 B1, ;
US 6562828 B1

146603-99-81-Boc-4-烯丙基-4-哌啶甲酸乙酯

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4427-25-22-氧杂-8-氮杂螺[4.5]癸烷-1-酮盐酸盐

参考文献

Cooper, Laura C.; Carlson, Emma J.; Castro, Jose L.; Chicchi, Gary G.; Dinnell, Kevin; Di Salvo, Jerry; Elliott, Jason M.; Hollingworth, Gregory J.; Kurtz, Marc M.; Ridgill, Mark P.; Rycroft, Wayne; Tsao, Kwei-Lan; Swain, Christopher J.
Bioorganic and Medicinal Chemistry Letters, 2002 , vol. 12, # 13 p. 1759 - 1762

146603-99-81-Boc-4-烯丙基-4-哌啶甲酸乙酯

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426842-70-81-Boc-4-烯丙基-4-哌啶甲酸

参考文献

Baque, Eric; Carry, Jean-Christophe; El-Ahmad, Youssef; Evers, Michel; Hubert, Philippe; Malleron, Jean-Luc; Mignani, Serge; Pantel, Guy; Tabart, Michel; Viviani, Fabrice
Patent: US2002/111492 A1, 2002 ;

146603-99-81-Boc-4-烯丙基-4-哌啶甲酸乙酯

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247133-32-04-(2-羟基乙基)-1,4-哌啶二羧酸 1-(1,1-二甲基乙基) 4-乙酯

参考文献

Cooper, Laura C.; Carlson, Emma J.; Castro, Jose L.; Chicchi, Gary G.; Dinnell, Kevin; Di Salvo, Jerry; Elliott, Jason M.; Hollingworth, Gregory J.; Kurtz, Marc M.; Ridgill, Mark P.; Rycroft, Wayne; Tsao, Kwei-Lan; Swain, Christopher J.
Bioorganic and Medicinal Chemistry Letters, 2002 , vol. 12, # 13 p. 1759 - 1762

146603-99-81-Boc-4-烯丙基-4-哌啶甲酸乙酯

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236406-38-54-(2-羟基乙基)-4-(羟基甲基)-1-哌啶羧酸 1,1-二甲基乙酯

参考文献

Cooper, Laura C.; Carlson, Emma J.; Castro, Jose L.; Chicchi, Gary G.; Dinnell, Kevin; Di Salvo, Jerry; Elliott, Jason M.; Hollingworth, Gregory J.; Kurtz, Marc M.; Ridgill, Mark P.; Rycroft, Wayne; Tsao, Kwei-Lan; Swain, Christopher J.
Bioorganic and Medicinal Chemistry Letters, 2002 , vol. 12, # 13 p. 1759 - 1762

146603-99-81-Boc-4-烯丙基-4-哌啶甲酸乙酯

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176-69-22-噁唑-8-氮杂螺[4.5]癸烷

参考文献

Cooper, Laura C.; Carlson, Emma J.; Castro, Jose L.; Chicchi, Gary G.; Dinnell, Kevin; Di Salvo, Jerry; Elliott, Jason M.; Hollingworth, Gregory J.; Kurtz, Marc M.; Ridgill, Mark P.; Rycroft, Wayne; Tsao, Kwei-Lan; Swain, Christopher J.
Bioorganic and Medicinal Chemistry Letters, 2002 , vol. 12, # 13 p. 1759 - 1762

146603-99-81-Boc-4-烯丙基-4-哌啶甲酸乙酯

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154348-08-01-氧代-2-噁-8-氮杂螺[4.5]癸烷-8-羧酸叔丁酯

参考文献

Pineiro, Jose Luis Castro; Dinnell, Kevin; Elliott, Jason Matthew; Hollingworth, Gregory John; Shaw, Duncan Edward; Swain, Christopher John; Yang, Lihu
Patent: US2003/225059 A1, 2003 ;
Location in patent: Page 27 ;