3,3-二甲基-[1,2,5]噻二唑烷 1,1-二氧化物合成路线 (共 2 条)
反应条件
pyridine 16.5 h; Heating / reflux;
参考文献
Bristol-Myers Squibb Company
Patent: US2008/9465 A1, 2008 ;
Location in patent: Page/Page column 97-98 ;
US 20080009465 A1
反应条件
amidosulfamic acid in pyridine 16 h;
参考文献
Castro, Jose L.; Baker, Raymond; Guiblin, Alexander R.; Hobbs, Sarah C.; Jenkins, Matthew; et al.
Journal of Medicinal Chemistry, 1994 , vol. 37, # 19 p. 3023 - 3032