2-(2-氯乙酰基氨基)-苯甲酸合成路线 （共 13 条）
反应条件
in benzene 2 h; Heating;
参考文献
Tetrahedron, , vol. 47, # 45 p. 9393 - 9410
反应条件
1.1: sodium hydroxide; bromine / water / 0.03 h / -5 °C / |Reflux 1.2: pH 4 - 5 2.1: N,N-dimethyl-formamide / 0 - 20 °C View Scheme
参考文献
Chemical Communications, , vol. 49, # 76 p. 8516 - 8518
参考文献
Indian Journal of Chemistry - Section B Organic and Medicinal Chemistry, , vol. 41, # 3 p. 647 - 649
参考文献
Yamato; Takeuchi; Chang; Hashigaki
Chemical and Pharmaceutical Bulletin, 1992 , vol. 40, # 2 p. 528 - 530
反应条件
phosphorus trichoride in toluene Condensation; 3 h; Heating;
参考文献
Farghaly; Moharram
Bollettino Chimico Farmaceutico, 1999 , vol. 138, # 6 p. 280 - 289
反应条件
phosphorus trichoride in toluene Condensation; 3 h; Heating;
参考文献
Farghaly; Moharram
Bollettino Chimico Farmaceutico, 1999 , vol. 138, # 6 p. 280 - 289
反应条件
1: 65 percent / POCl3 / toluene / 115 °C 2: 90 percent / NaN3 / dimethylformamide / 2 h / Ambient temperature 3: 83 percent / H2S / pyridine; H2O / 1.5 h / Ambient temperature View Scheme
参考文献
Domanig, Rainer
Monatshefte fuer Chemie, 1981 , vol. 112, p. 1195 - 1202
反应条件
1: in toluene T=20°C; 0.5 h; 2: With trichlorophosphate in toluene Heating / reflux;
参考文献
Giri, Rajan S.; Thaker, Hardik M.; Giordano, Tony; Williams, Jill; Rogers, Donna; Vasu, Kamala K.; Sudarsanam, Vasudevan
Bioorganic and Medicinal Chemistry, 2010 , vol. 18, # 7 p. 2796 - 2808
参考文献
Mect Corporation
Patent: US5217961 A1, 1993 ;
反应条件
1: 18 percent / DMF / DMAP / 80 - 90 °C
2: 36 percent / PPS / 2 h / 120 °C
View Scheme
参考文献
Goerlitzer; Weber
Archiv der Pharmazie, 1981 , vol. 314, # 10 p. 852 - 861
