反应条件
sodium hydride in N,N-dimethyl-formamide
1.) 30 deg C, 2h, 2.) 50-55 deg C, 4h;
参考文献
Glushkov, R. G.; Vasil'evykh, L. G.; Kogan, Z. S.; Gorkin, V. Z.
Pharmaceutical Chemistry Journal, 1981 , vol. 15, # 5 p. 337 - 341
Khimiko-Farmatsevticheskii Zhurnal, 1981 , vol. 15, # 5 p. 58 - 62