反应条件
1: SOCl2, Py / toluene; dimethylformamide / 0.08 h / 0 °C 2: Et3N, DMAP / CH2Cl2 / Ambient temperature View Scheme
参考文献
Pacofsky, Gregory J.; Lackey, Karen; Alligood, Krystal J.; Berman, Judd; Charifson, Paul S.; Crosby, Renae M.; Dorsey Jr., George F.; Feldman, Paul L.; Gilmer, Tona M.; Hummel, Conrad W.; Jordan, Steven R.; Mohr, Christopher; Shewchuk, Lisa M.; Sternbach, Daniel D.; Rodriguez, Marc
Journal of Medicinal Chemistry, 1998 , vol. 41, # 11 p. 1894 - 1908