反应条件
1: imidazole / dimethylformamide / 1.75 h 2: 1.) H2O, AcOH; 2.) N,N-dimethylolpyridine / 1.) methanol, toluene, r.t., 1 h; 2) ether, 1 h 3: 80 percent / tetra-n-butylammonium fluoride / tetrahydrofuran / 0.5 h / 5 °C 4: 90 percent / aq.NaOH / methanol / 2.5 h / 5 - 25 °C View Scheme
参考文献
Canadian Journal of Chemistry, , vol. 62, p. 1169 - 1175