1-异氰酰基-2-苯磺酰基苯合成路线 (共 3 条)
反应条件
in 1,4-dioxane T=20 - 60°C; 1 h;
参考文献
ELI LILLY AND COMPANY
Patent: WO2005/26177 A1, 2005 ;
Location in patent: Page/Page column 75 ;
WO 2005/026177 A1
参考文献
Schmutz,J. et al.
Helvetica Chimica Acta, 1965 , vol. 48, p. 336 - 347
反应条件
AlCl3, aluminium chloride in 1,2-dichloro-benzene T=100 - 150°C; 4 h;
参考文献
ELI LILLY AND COMPANY
Patent: WO2005/26177 A1, 2005 ;
Location in patent: Page/Page column 75 ;
WO 2005/026177 A1