3,5-二(叔-丁基二甲基硅烷基)罗舒伐他汀合成路线 (共 2 条)
反应条件
lithium hydroxide hydrate in methanol T=20°C; 12 h;
参考文献
NICOX S.A.; STORONI, Laura; BONFANTI, Annalisa; BENEDINI, Francesca; OLIVA, Francesca; MIGLIETTA, Daniela; ONGINI, Ennio
Patent: WO2011/160974 A2, 2011 ;
Location in patent: Page/Page column 60-61 ;
反应条件
1: 1H-imidazole / N,N-dimethyl-formamide / 12 h / 20 °C 2: lithium hydroxide hydrate / methanol / 12 h / 20 °C View Scheme
参考文献
NICOX S.A.; STORONI, Laura; BONFANTI, Annalisa; BENEDINI, Francesca; OLIVA, Francesca; MIGLIETTA, Daniela; ONGINI, Ennio
Patent: WO2011/160974 A2, 2011 ;