1: With dimethylsulfide borane complex in tetrahydrofuran T=0 - 20°C; 12.5 h; 2: With hydrogenchloride; methanol; water in tetrahydrofuran 3: With water; sodium hydrogencarbonate
参考文献
BRISTOL-MYERS SQUIBB COMPANY
Patent: WO2008/79759 A1, 2008 ;
Location in patent: Page/Page column 125 ;
WO 2008/079759 A1